High-affinity fluorescent ligands for the 5-HT3 receptor
نویسندگان
چکیده
منابع مشابه
High-affinity fluorescent ligands for the 5-HT3 receptor
The synthesis, photophysical and biological characterization of a small library of fluorescent 5-HT(3) receptor ligands is described. Several of these novel granisetron conjugates have high quantum yields and show high affinity for the human 5-HT(3)AR.
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ژورنال
عنوان ژورنال: Bioorganic & Medicinal Chemistry Letters
سال: 2012
ISSN: 0960-894X
DOI: 10.1016/j.bmcl.2011.11.097